Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules
Por um escritor misterioso
Last updated 06 julho 2024
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Identification of Protein Substrates of Specific PARP Enzymes Using Analog-Sensitive PARP Mutants and a Clickable NAD+ Analog. - Abstract - Europe PMC
![Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules](https://pubs.acs.org/cms/10.1021/acs.jmedchem.2c00281/asset/images/large/jm2c00281_0024.jpeg)
Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules
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ADP-ribose contributions to genome stability and PARP enzyme trapping on sites of DNA damage; paradigm shifts for a coming-of-age modification - Journal of Biological Chemistry
![Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules](https://www.pnas.org/cms/10.1073/pnas.2121979119/asset/f95f6865-fc6f-45b1-bc74-466d2cc3f1bc/assets/images/large/pnas.2121979119fig01.jpg)
Inhibitors of PARP: Number crunching and structure gazing
![Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules](https://d3i71xaburhd42.cloudfront.net/2036d76bc2799cb7acf75d040809fd12060e4497/6-Figure4-1.png)
PDF] Enabling drug discovery for the PARP protein family through the detection of mono-ADP-ribosylation.
![Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules](https://www.frontiersin.org/files/Articles/811671/fmicb-12-811671-HTML/image_m/fmicb-12-811671-g001.jpg)
Frontiers Virus–Host Interplay Between Poly (ADP-Ribose) Polymerase 1 and Oncogenic Gammaherpesviruses
![Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules](https://d3i71xaburhd42.cloudfront.net/2036d76bc2799cb7acf75d040809fd12060e4497/3-Figure1-1.png)
PDF] Enabling drug discovery for the PARP protein family through the detection of mono-ADP-ribosylation.
![Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules](https://media.springernature.com/m685/springer-static/image/art%3A10.1007%2Fs00018-022-04290-6/MediaObjects/18_2022_4290_Fig3_HTML.png)
Intracellular mono-ADP-ribosyltransferases at the host–virus interphase
![Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules](https://pubs.acs.org/cms/10.1021/acs.jmedchem.2c00281/asset/images/large/jm2c00281_0012.jpeg)
Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules
![Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules](https://pubs.acs.org/cms/10.1021/acs.jmedchem.2c00281/asset/images/medium/jm2c00281_0013.gif)
Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules
![Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules](https://pubs.acs.org/cms/10.1021/acs.jmedchem.2c00281/asset/images/medium/jm2c00281_0023.gif)
Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules
![Medicinal Chemistry Perspective on Targeting Mono-ADP-Ribosylating PARPs with Small Molecules](https://www.mdpi.com/molecules/molecules-28-05849/article_deploy/html/images/molecules-28-05849-g008.png)
Molecules, Free Full-Text
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Intracellular mono-ADP-ribosyltransferases at the host–virus interphase
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